Synthesis, herbicidal activity, and structure-bioactivity relationship of pyridyl-containing 2-phenyliminothiazolidines

Gangyue Li; Xuhong Qian; Shenggang Yan; Jingnan Cui; Rong Zhang; Yi Xiao

doi:10.1007/s00706-007-0696-0

Synthesis, herbicidal activity, and structure-bioactivity relationship of pyridyl-containing 2-phenyliminothiazolidines

Gangyue Li
, Xuhong Qian^*
, Shenggang Yan
, Jingnan Cui
, Rong Zhang
, Yi Xiao

^*此作品的通讯作者

Dalian Maritime University
Dalian University of Technology
East China University of Science and Technology

科研成果: 期刊稿件 › 文章 › 同行评审

3 引用（Scopus）

摘要

A series of novel 2-phenyliminothiazolidine derivatives were designed and synthesized. All title compounds were characterized by ¹H NMR and, in some cases, by ¹³C NMR, IR, and HRMS. Their agricultural bioactivities were evaluated and some of these compounds exhibited efficient herbicidal activities against Echinochloa crusgalli, Sorghum vulgare, Digitaria sanguinalis, Eclipta prostrasta, Cucumis sativus, and Brassica campestris at 50∈μg/cm³. Analysis of the quantitative structure-activity relationship (QSAR) showed that the electronic parameter was the main factor to affect herbicidal activities.

源语言	英语
页（从-至）	169-178
页数	10
期刊	Monatshefte fur Chemie
卷	139
期	2
DOI	https://doi.org/10.1007/s00706-007-0696-0
出版状态	已出版 - 2月 2008
已对外发布	是

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abstract = "A series of novel 2-phenyliminothiazolidine derivatives were designed and synthesized. All title compounds were characterized by 1H NMR and, in some cases, by 13C NMR, IR, and HRMS. Their agricultural bioactivities were evaluated and some of these compounds exhibited efficient herbicidal activities against Echinochloa crusgalli, Sorghum vulgare, Digitaria sanguinalis, Eclipta prostrasta, Cucumis sativus, and Brassica campestris at 50∈μg/cm3. Analysis of the quantitative structure-activity relationship (QSAR) showed that the electronic parameter was the main factor to affect herbicidal activities.",

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author = "Gangyue Li and Xuhong Qian and Shenggang Yan and Jingnan Cui and Rong Zhang and Yi Xiao",

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doi = "10.1007/s00706-007-0696-0",

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T1 - Synthesis, herbicidal activity, and structure-bioactivity relationship of pyridyl-containing 2-phenyliminothiazolidines

AU - Li, Gangyue

AU - Qian, Xuhong

AU - Yan, Shenggang

AU - Cui, Jingnan

AU - Zhang, Rong

AU - Xiao, Yi

PY - 2008/2

Y1 - 2008/2

N2 - A series of novel 2-phenyliminothiazolidine derivatives were designed and synthesized. All title compounds were characterized by 1H NMR and, in some cases, by 13C NMR, IR, and HRMS. Their agricultural bioactivities were evaluated and some of these compounds exhibited efficient herbicidal activities against Echinochloa crusgalli, Sorghum vulgare, Digitaria sanguinalis, Eclipta prostrasta, Cucumis sativus, and Brassica campestris at 50∈μg/cm3. Analysis of the quantitative structure-activity relationship (QSAR) showed that the electronic parameter was the main factor to affect herbicidal activities.

AB - A series of novel 2-phenyliminothiazolidine derivatives were designed and synthesized. All title compounds were characterized by 1H NMR and, in some cases, by 13C NMR, IR, and HRMS. Their agricultural bioactivities were evaluated and some of these compounds exhibited efficient herbicidal activities against Echinochloa crusgalli, Sorghum vulgare, Digitaria sanguinalis, Eclipta prostrasta, Cucumis sativus, and Brassica campestris at 50∈μg/cm3. Analysis of the quantitative structure-activity relationship (QSAR) showed that the electronic parameter was the main factor to affect herbicidal activities.

KW - 2-Phenyliminothiazolidine

KW - Herbicidal activity

KW - QSAR

KW - Synthesis

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U2 - 10.1007/s00706-007-0696-0

DO - 10.1007/s00706-007-0696-0

M3 - 文章

AN - SCOPUS:38949168961

SN - 0026-9247

VL - 139

SP - 169

EP - 178

JO - Monatshefte fur Chemie

JF - Monatshefte fur Chemie

IS - 2

ER -

Synthesis, herbicidal activity, and structure-bioactivity relationship of pyridyl-containing 2-phenyliminothiazolidines

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