TY - JOUR
T1 - Synthesis, herbicidal activity, and structure-bioactivity relationship of pyridyl-containing 2-phenyliminothiazolidines
AU - Li, Gangyue
AU - Qian, Xuhong
AU - Yan, Shenggang
AU - Cui, Jingnan
AU - Zhang, Rong
AU - Xiao, Yi
PY - 2008/2
Y1 - 2008/2
N2 - A series of novel 2-phenyliminothiazolidine derivatives were designed and synthesized. All title compounds were characterized by 1H NMR and, in some cases, by 13C NMR, IR, and HRMS. Their agricultural bioactivities were evaluated and some of these compounds exhibited efficient herbicidal activities against Echinochloa crusgalli, Sorghum vulgare, Digitaria sanguinalis, Eclipta prostrasta, Cucumis sativus, and Brassica campestris at 50∈μg/cm3. Analysis of the quantitative structure-activity relationship (QSAR) showed that the electronic parameter was the main factor to affect herbicidal activities.
AB - A series of novel 2-phenyliminothiazolidine derivatives were designed and synthesized. All title compounds were characterized by 1H NMR and, in some cases, by 13C NMR, IR, and HRMS. Their agricultural bioactivities were evaluated and some of these compounds exhibited efficient herbicidal activities against Echinochloa crusgalli, Sorghum vulgare, Digitaria sanguinalis, Eclipta prostrasta, Cucumis sativus, and Brassica campestris at 50∈μg/cm3. Analysis of the quantitative structure-activity relationship (QSAR) showed that the electronic parameter was the main factor to affect herbicidal activities.
KW - 2-Phenyliminothiazolidine
KW - Herbicidal activity
KW - QSAR
KW - Synthesis
UR - https://www.scopus.com/pages/publications/38949168961
U2 - 10.1007/s00706-007-0696-0
DO - 10.1007/s00706-007-0696-0
M3 - 文章
AN - SCOPUS:38949168961
SN - 0026-9247
VL - 139
SP - 169
EP - 178
JO - Monatshefte fur Chemie
JF - Monatshefte fur Chemie
IS - 2
ER -