Pd-Catalyzed C-H/N-H Arylation: One-Pot Synthesis of Indolo[1, 2-f]phenanthridines

Lingkai Kong; Qiyi Yao; Mengdan Wang; Ruizhuo Sun; Yanzhong Li

doi:10.1002/slct.201701939

Pd-Catalyzed C-H/N-H Arylation: One-Pot Synthesis of Indolo[1, 2-f]phenanthridines

Lingkai Kong
, Qiyi Yao
, Mengdan Wang
, Ruizhuo Sun
, Yanzhong Li^*

^*Corresponding author for this work

School of Chemistry and Molecular Engineering

East China Normal University

Research output: Contribution to journal › Article › peer-review

11 Scopus citations

Abstract

A novel Pd-catalyzed method for the synthesis of indolo[1, 2-f]phenanthridines from 2-bromo-2′-iodo-1,1′-biphenyl and indole derivatives has been reported. The reaction involves direct N−H and C2-H arylation of indole. This Pd-catalyzed double arylation provides a useful route to synthesize indolo[1, 2-f]phenanthridine derivatives from simple and readily accessible starting materials.

Original language	English
Pages (from-to)	456-460
Number of pages	5
Journal	ChemistrySelect
Volume	3
Issue number	2
DOIs	https://doi.org/10.1002/slct.201701939
State	Published - 17 Jan 2018

Keywords

2-Bromo-2′-iodo-1,1′-biphenyl
C−H activation
Indolo[1, 2-f]phenanthridines
palladium catalysis

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10.1002/slct.201701939

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title = "Pd-Catalyzed C-H/N-H Arylation: One-Pot Synthesis of Indolo[1, 2-f]phenanthridines",

abstract = "A novel Pd-catalyzed method for the synthesis of indolo[1, 2-f]phenanthridines from 2-bromo-2′-iodo-1,1′-biphenyl and indole derivatives has been reported. The reaction involves direct N−H and C2-H arylation of indole. This Pd-catalyzed double arylation provides a useful route to synthesize indolo[1, 2-f]phenanthridine derivatives from simple and readily accessible starting materials.",

keywords = "2-Bromo-2′-iodo-1,1′-biphenyl, C−H activation, Indolo[1, 2-f]phenanthridines, palladium catalysis",

author = "Lingkai Kong and Qiyi Yao and Mengdan Wang and Ruizhuo Sun and Yanzhong Li",

note = "Publisher Copyright: {\textcopyright} 2018 Wiley-VCH Verlag GmbH \& Co. KGaA, Weinheim",

year = "2018",

month = jan,

day = "17",

doi = "10.1002/slct.201701939",

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TY - JOUR

T1 - Pd-Catalyzed C-H/N-H Arylation

T2 - One-Pot Synthesis of Indolo[1, 2-f]phenanthridines

AU - Kong, Lingkai

AU - Yao, Qiyi

AU - Wang, Mengdan

AU - Sun, Ruizhuo

AU - Li, Yanzhong

PY - 2018/1/17

Y1 - 2018/1/17

N2 - A novel Pd-catalyzed method for the synthesis of indolo[1, 2-f]phenanthridines from 2-bromo-2′-iodo-1,1′-biphenyl and indole derivatives has been reported. The reaction involves direct N−H and C2-H arylation of indole. This Pd-catalyzed double arylation provides a useful route to synthesize indolo[1, 2-f]phenanthridine derivatives from simple and readily accessible starting materials.

AB - A novel Pd-catalyzed method for the synthesis of indolo[1, 2-f]phenanthridines from 2-bromo-2′-iodo-1,1′-biphenyl and indole derivatives has been reported. The reaction involves direct N−H and C2-H arylation of indole. This Pd-catalyzed double arylation provides a useful route to synthesize indolo[1, 2-f]phenanthridine derivatives from simple and readily accessible starting materials.

KW - 2-Bromo-2′-iodo-1,1′-biphenyl

KW - C−H activation

KW - Indolo[1, 2-f]phenanthridines

KW - palladium catalysis

UR - https://www.scopus.com/pages/publications/85044256659

U2 - 10.1002/slct.201701939

DO - 10.1002/slct.201701939

M3 - 文章

AN - SCOPUS:85044256659

SN - 2365-6549

VL - 3

SP - 456

EP - 460

JO - ChemistrySelect

JF - ChemistrySelect

IS - 2

ER -

Pd-Catalyzed C-H/N-H Arylation: One-Pot Synthesis of Indolo[1, 2-f]phenanthridines

Abstract

Keywords

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