An efficient and practical method for the synthesis of 1-(2,6- difluorobenzoyl)-3-(2-alkyl-3-oxopyridazin-4-yl)ureas as potential chitin synthesis inhibitors

Song Cao; De Li Lu; Chuan Meng Zhao; Li Na Li; Qing Chun Huang; Xu Hong Qian

doi:10.1007/s00706-005-0476-7

An efficient and practical method for the synthesis of 1-(2,6- difluorobenzoyl)-3-(2-alkyl-3-oxopyridazin-4-yl)ureas as potential chitin synthesis inhibitors

Song Cao
, De Li Lu
, Chuan Meng Zhao
, Li Na Li
, Qing Chun Huang
, Xu Hong Qian

Unknown

Research output: Contribution to journal › Article › peer-review

8 Scopus citations

Abstract

A mild and efficient method for the synthesis of 4-amino-3(2H)- pyridazinones from their corresponding 4,5-dichloropyridazinones under microwave-assisted conditions is described. A series of novel chitin synthesis inhibitors, benzoylphenylureas containing the 3(2H)-pyridazinone, were synthesized. The biological activity of these target compounds was evaluated.

Original language	English
Pages (from-to)	779-784
Number of pages	6
Journal	Monatshefte fur Chemie
Volume	137
Issue number	6
DOIs	https://doi.org/10.1007/s00706-005-0476-7
State	Published - Jun 2006
Externally published	Yes

Keywords

Bioorganic chemistry
Heterocycles
Insecticidal activity
Microwave

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10.1007/s00706-005-0476-7

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title = "An efficient and practical method for the synthesis of 1-(2,6- difluorobenzoyl)-3-(2-alkyl-3-oxopyridazin-4-yl)ureas as potential chitin synthesis inhibitors",

abstract = "A mild and efficient method for the synthesis of 4-amino-3(2H)- pyridazinones from their corresponding 4,5-dichloropyridazinones under microwave-assisted conditions is described. A series of novel chitin synthesis inhibitors, benzoylphenylureas containing the 3(2H)-pyridazinone, were synthesized. The biological activity of these target compounds was evaluated.",

keywords = "Bioorganic chemistry, Heterocycles, Insecticidal activity, Microwave",

author = "Song Cao and Lu, \{De Li\} and Zhao, \{Chuan Meng\} and Li, \{Li Na\} and Huang, \{Qing Chun\} and Qian, \{Xu Hong\}",

year = "2006",

month = jun,

doi = "10.1007/s00706-005-0476-7",

language = "英语",

volume = "137",

pages = "779--784",

journal = "Monatshefte fur Chemie",

issn = "0026-9247",

publisher = "Springer",

number = "6",

}

TY - JOUR

T1 - An efficient and practical method for the synthesis of 1-(2,6- difluorobenzoyl)-3-(2-alkyl-3-oxopyridazin-4-yl)ureas as potential chitin synthesis inhibitors

AU - Cao, Song

AU - Lu, De Li

AU - Zhao, Chuan Meng

AU - Li, Li Na

AU - Huang, Qing Chun

AU - Qian, Xu Hong

PY - 2006/6

Y1 - 2006/6

N2 - A mild and efficient method for the synthesis of 4-amino-3(2H)- pyridazinones from their corresponding 4,5-dichloropyridazinones under microwave-assisted conditions is described. A series of novel chitin synthesis inhibitors, benzoylphenylureas containing the 3(2H)-pyridazinone, were synthesized. The biological activity of these target compounds was evaluated.

AB - A mild and efficient method for the synthesis of 4-amino-3(2H)- pyridazinones from their corresponding 4,5-dichloropyridazinones under microwave-assisted conditions is described. A series of novel chitin synthesis inhibitors, benzoylphenylureas containing the 3(2H)-pyridazinone, were synthesized. The biological activity of these target compounds was evaluated.

KW - Bioorganic chemistry

KW - Heterocycles

KW - Insecticidal activity

KW - Microwave

UR - https://www.scopus.com/pages/publications/33745025736

U2 - 10.1007/s00706-005-0476-7

DO - 10.1007/s00706-005-0476-7

M3 - 文章

AN - SCOPUS:33745025736

SN - 0026-9247

VL - 137

SP - 779

EP - 784

JO - Monatshefte fur Chemie

JF - Monatshefte fur Chemie

IS - 6

ER -

An efficient and practical method for the synthesis of 1-(2,6- difluorobenzoyl)-3-(2-alkyl-3-oxopyridazin-4-yl)ureas as potential chitin synthesis inhibitors

Abstract

Keywords

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